Triptorelin is a gonadotropin-releasing hormone (GnRH) agonist used to treat hormone-sensitive conditions such as advanced prostate cancer, endometriosis, and precocious puberty.
1 Box – 10 vials
$338.00
Triptorelin is a gonadotropin-releasing hormone (GnRH) agonist used to treat hormone-sensitive conditions such as advanced prostate cancer, endometriosis, and precocious puberty.
1 Box – 10 vials
Triptorelin is a gonadotropin releasing hormone analogue that has been used in the clinical setting to treat advanced prostate cancer as part of a multi-faceted approach to androgen deprivation therapy. Similar to luteinizing hormone releasing hormone, triptorelin is a potent inhibitor of testosterone and estrogen synthesis when given in long-term, continuous dosing. In the UK, triptorelin is used to suppress testosterone and estrogen synthesis in transgender people. The peptide has also found application in the treatment of hormone-receptor positive breast cancer in premenopausal women.
Triptorelin Restores Testosterone Secretion in Some Men
The way in which triptorelin is used can dramatically change the effects that the peptide has. Research has shown that triptorelin increases testosterone levels early during prolonged treatment regiments and only begins to suppress production after chronic exposure to the peptide. This is referred to as testosterone flare and is seen in the first few weeks of triptorelin treatment. This suggests that triptorelin may be useful in boosting testosterone levels in some men if administered with appropriate timing and in appropriate doses.
Triptorelin Administration Determines Effects
Triptorelin is an analogue of gonadotropin releasing hormone (GnRH). As such, it can stimulate the anterior pituitary gland to release follicle-stimulating hormone (FSH) and luteinizing hormone (LH). If given in a pulsatile manner, this is precisely what triptorelin does. Exact levels of FSH and LH depend on the size and frequency of GnRH pulses and thus on the size and frequency of triptorelin dosing. If, however, triptorelin is given in a steady-state format rather than in a pulsatile manner, it will eventually suppress LH and FSH secretion as well as the production of testosterone and estrogen. How triptorelin is administered in research settings will determine what its ultimate properties are.
Product name | Triptorelin Acetate/GnRH Triptorelin | ![]() |
CAS NO | 140194-24-7 | |
Quantity | 2mg | |
Batch NO | OP-10213C |
All of our products are manufactured using the Lyophilization (Freeze Drying) process, which ensures that our products remain 100% stable for shipping for up to 3-4 months.
Once the peptides are reconstituted (mixed with bacteriostatic water), they must be stored in the fridge to maintain stability. After reconstitution, the peptides will remain stable for up to 30 days.
Lyophilization is a unique dehydration process, also known as cryodesiccation, where the peptides are frozen and then subjected to low pressure. This causes the water in the peptide vial to sublimate directly from solid to gas, leaving behind a stable, crystalline white structure known as lyophilized peptide. The puffy white powder can be stored at room temperature until you’re ready to reconstitute it with bacteriostatic water.
Once peptides have been received, it is imperative that they are kept cold and away from light. If the peptides will be used immediately, or in the next several days, weeks or months, short-term refrigeration under 4C (39F) is generally acceptable. Lyophilized peptides are usually stable at room temperatures for several weeks or more, so if they will be utilized within weeks or months such storage is typically adequate.
However, for longer term storage (several months to years) it is more preferable to store peptides in a freezer at -80C (-112F). When storing peptides for months or even years, freezing is optimal in order to preserve the peptide’s stability.
Specification | 2mg*10vials |
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